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100 _aGirish Meravanige1
245 _aDesign and Development of Anti-fungal Topical Gel Loaded with Solid Lipid Nanoparticles for Wound Healing
300 _ap122-130
520 _aThe topical administration of anti-fungal drugs by Solid Lipid Nanoparticles (SLNs) has enormous potential. This study aimed to develop a topical 5-flucytosine-loaded SLNs gel to improve the efficacy of the well-known anti-fungal drug in the treatment of wound healing. Materials and Methods: In order to create 5-flucytosine SLNs, a five-level, two-factor Central-composite design was used. Stearic acid and Poloxamer 407 concentrations of surfactants were chosen as independent factors, and particle size and %Entrapment Efficiency (%EE) were chosen as dependent variables. The produced 5-Flucytosine-SLNs were examined using SEM analysis, zeta potential, polydispersity index, and particle size measurements. Additionally, Carbopol 934 was used to incorporate the improved 5-Flucytosine-SLN formula into gel. Results: The outcomes demonstrated that 5-Flucytosine-SLNs had colloidal sizes with an essentially spherical shape and no aggregation. 5-Flucytosine-SLNs were discovered to have a particle size of 720.4 nm and an Entrapment Efficiency (EE) of 90.28%. The in vitro release, among other assessment criteria, was evaluated for the improved SLN gels. Conclusion: The study's conclusions imply that the topical gels made with 5-Flucytosine-loaded SLNs must be effective in the management of wound healing.
654 _a 5-Flucytosine
_aSolid lipid nanoparticle
_aCentral-composite design
_aTopical delivery,
_a Optimization.
700 _aRanjitha B2
_aPrakash Goudanavar2
_aGSN Koteswara Rao3
_aB Nirmala Devi4
_a N. Raghavendra Naveen2,
_a Afzal Haq Asif5
_a Sree Harsha Nagaraja6,7
_a Mohammed Monirul Islam8
_aPavan Kumar
_aPavagada Sreenivasalu9,
_a, Mallikarjun Telsang10
_a, Krishna Swaroop Duddi Sreehari1
773 0 _0125266
_9109601
_dBanglore Association of Pharmaceutical Tearchers of India
_oJP44
_tIndian Journal of Pharmaceutical Education and Research
_x0019-5464
942 _cJA
942 _2ddc
999 _c130064
_d130064